Apelin Receptor Signaling and Biased Agonism

This paper identifies (-)-epicatechin as a biased ligand of the apelin receptor, supporting a receptor-mediated signaling mechanism that may help explain some of its vascular and metabolic effects.

This paper identifies (-)-epicatechin as a biased ligand of the apelin receptor, supporting a receptor-mediated signaling mechanism that may help explain some of its vascular and metabolic effects.